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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Epizyme

US Patent
LigandPNGBDBM440046(US10633389, Example 384-1a | US20230279020, Exampl...)
Affinity DataIC50:  550nMAssay Description:The assays were all performed in a buffer consisting of 20 mM Bicine (pH=7.6), 1 mM TCEP, 0.005% BSG, and 0.002% Tween 20, prepared on the day of use...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Epizyme

US Patent
LigandPNGBDBM440046(US10633389, Example 384-1a | US20230279020, Exampl...)
Affinity DataIC50:  550nMAssay Description:The assays were all performed in a buffer consisting of 20 mM Bicine (pH=7.6), 1 mM TCEP, 0.005% BSG, and 0.002% Tween 20, prepared on the day of use...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent