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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Cystic fibrosis transmembrane conductance regulator
(Homo sapiens (Human))
University Of California
Curated by
ChEMBL
Ligand
BDBM50232962
(CHEMBL4079174)
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Affinity Data
EC50: 31nM
Assay Description:
Activation of human CFTR expressed in forskolin-stimulated basolateral membrane permeabilized FRT cells co-expressing YFP assessed as increase in sho...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Cystic fibrosis transmembrane conductance regulator
(Homo sapiens (Human))
University Of California
Curated by
ChEMBL
Ligand
BDBM50232962
(CHEMBL4079174)
Copy SMILES
Copy InChI
Affinity Data
EC50: 40nM
Assay Description:
Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI