Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetStromelysin-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50131663(3-{1-[(Methoxy-phenyl-methyl)-carbamoyl]-2,2-dimet...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human matrix metalloprotease-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50131663(3-{1-[(Methoxy-phenyl-methyl)-carbamoyl]-2,2-dimet...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50131663(3-{1-[(Methoxy-phenyl-methyl)-carbamoyl]-2,2-dimet...)
Affinity DataIC50:  3.04E+4nMAssay Description:Inhibition of human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50131663(3-{1-[(Methoxy-phenyl-methyl)-carbamoyl]-2,2-dimet...)
Affinity DataIC50:  3.42E+4nMAssay Description:Inhibition of human matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50131663(3-{1-[(Methoxy-phenyl-methyl)-carbamoyl]-2,2-dimet...)
Affinity DataIC50:  6.69E+4nMAssay Description:Inhibition of Matrix metalloprotease-14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed