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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Aeovian Pharmaceuticals

US Patent
LigandPNGBDBM597720(US11603377, Compound 41)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Aeovian Pharmaceuticals

US Patent
LigandPNGBDBM597720(US11603377, Compound 41)
Affinity DataKd: >800nMAssay Description:Biotinylated avi-FKBP51 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Aeovian Pharmaceuticals

US Patent
LigandPNGBDBM597720(US11603377, Compound 41)
Affinity DataKd: >800nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Aeovian Pharmaceuticals

US Patent
LigandPNGBDBM597720(US11603377, Compound 41)
Affinity DataKd: >100nMAssay Description:Biotinylated avi-FKBP51 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent