Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAminopeptidase N(Sus scrofa (Pig))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL

LigandBDBM50001944(2-(3,7-Diamino-2-hydroxy-heptanoylamino)-3-[2-(2-n...)Copy SMILESCopy InChI

Affinity DataIC50:  3.27E+4nMAssay Description:Inhibitory potency against purified membrane bound rat brain aminopeptidaseMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetAminopeptidase B(Rattus norvegicus)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL

LigandBDBM50001944(2-(3,7-Diamino-2-hydroxy-heptanoylamino)-3-[2-(2-n...)Copy SMILESCopy InChI

Affinity DataIC50:  5.83E+5nMAssay Description:Inhibitory potency against purified membrane bound rat brain Aminopeptidase B (AP-B) using L-lysine-beta napthylamide as substrateMore data for this Ligand-Target Pair

Target InfoKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetAminopeptidase N(Rattus norvegicus)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL

LigandBDBM50001944(2-(3,7-Diamino-2-hydroxy-heptanoylamino)-3-[2-(2-n...)Copy SMILESCopy InChI

Affinity DataIC50:  8.52E+5nMAssay Description:Inhibitory potency against purified membrane bound rat brain Aminopeptidase M (AP-M) using [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair

Target InfoReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI