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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Dual specificity tyrosine-phosphorylation-regulated kinase 2
(Homo sapiens (Human))
University Of Athens
Curated by
ChEMBL
Ligand
BDBM50426322
(CHEMBL2321953)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human recombinant GST-fused DYRK2 expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counti...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(RAT)
University Of Athens
Curated by
ChEMBL
Ligand
BDBM50426322
(CHEMBL2321953)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Cyclin-dependent kinase 5
(Homo sapiens (Human))
University Of Athens
Curated by
ChEMBL
Ligand
BDBM50426322
(CHEMBL2321953)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human recombinant CDK5
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Glycogen synthase kinase-3 beta
(Sus scrofa)
University Of Athens
Curated by
ChEMBL
Ligand
BDBM50426322
(CHEMBL2321953)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of porcine brain GSK3beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/TrEMBL
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Casein kinase I isoform alpha
(Sus scrofa)
University Of Athens
Curated by
ChEMBL
Ligand
BDBM50426322
(CHEMBL2321953)
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Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of porcine brain CK1 using RRKHAAIGpSAYSITA as substrate
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI