Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426322(CHEMBL2321953)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant GST-fused DYRK2 expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50426322(CHEMBL2321953)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426322(CHEMBL2321953)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426322(CHEMBL2321953)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of porcine brain GSK3beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426322(CHEMBL2321953)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of porcine brain CK1 using RRKHAAIGpSAYSITA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed