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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM50434340
(CHEMBL2386760 | US9446044, 89)
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Affinity Data
IC50: 5.10nM
Assay Description:
Inhibition of recombinant DYRK1A (unknown origin) after 120 mins in presence of [33P]-ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM50434340
(CHEMBL2386760 | US9446044, 89)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.10nM
pH: 7.5 T: 2°C
Assay Description:
The DYRK1A and DYRK1B kinase assays to determine IC50 values were performed by Reaction Biology Corporation using HotSpot technology Worldwide websit...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Dual specificity tyrosine-phosphorylation-regulated kinase 1B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM50434340
(CHEMBL2386760 | US9446044, 89)
Copy SMILES
Copy InChI
Affinity Data
IC50: 7.70nM
Assay Description:
Inhibition of recombinant DYRK1B (unknown origin) after 120 mins in presence of [33P]-ATP
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Dual specificity tyrosine-phosphorylation-regulated kinase 1B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM50434340
(CHEMBL2386760 | US9446044, 89)
Copy SMILES
Copy InChI
Affinity Data
IC50: 7.70nM
pH: 7.5 T: 2°C
Assay Description:
The DYRK1A and DYRK1B kinase assays to determine IC50 values were performed by Reaction Biology Corporation using HotSpot technology Worldwide websit...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI