Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 10 hits in this display
Caspase-3(Homo sapiens (Human))University Hospital Of The WestfäLische Wilhelms-UniversitäT
Curated by ChEMBL
BDBM50200302((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Caspase-3(Homo sapiens (Human))University Hospital Of The WestfäLische Wilhelms-UniversitäT
Curated by ChEMBL
BDBM50200302((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Caspase-3(Homo sapiens (Human))University Hospital Of The WestfäLische Wilhelms-UniversitäT
Curated by ChEMBL
BDBM50200302((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
IC50: 2.40nMAssay Description:Inhibition of human recombinant caspase 3 using Ac-DEVD-AMC substrate assessed as accumulation of cleaved fluorogenic productMore data for this Ligand-Target Pair
Caspase-3(Homo sapiens (Human))University Hospital Of The WestfäLische Wilhelms-UniversitäT
Curated by ChEMBL
BDBM50200302((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Caspase-7(Homo sapiens (Human))WestfäLische Wilhelms-UniversitäT
Curated by ChEMBL
BDBM50200302((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Caspase-7(Homo sapiens (Human))WestfäLische Wilhelms-UniversitäT
Curated by ChEMBL
BDBM50200302((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
IC50: 304nMAssay Description:Inhibition of human recombinant caspase 7 using Ac-DEVD-AMC substrate assessed as accumulation of cleaved fluorogenic productMore data for this Ligand-Target Pair
Caspase-7(Homo sapiens (Human))WestfäLische Wilhelms-UniversitäT
Curated by ChEMBL
BDBM50200302((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Caspase-1(Homo sapiens (Human))University Hospital Of The WestfäLische Wilhelms-UniversitäT
Curated by ChEMBL
BDBM50200302((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Caspase-6(Homo sapiens (Human))University Hospital Of The WestfäLische Wilhelms-UniversitäT
Curated by ChEMBL
BDBM50200302((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Caspase-8(Homo sapiens (Human))University Hospital Of The WestfäLische Wilhelms-UniversitäT
Curated by ChEMBL
BDBM50200302((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)