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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetCollagenase 3(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50265076((R)-2-(4'-((5-bromo-4-methoxy-3-methylbenzofuran-2...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50265076((R)-2-(4'-((5-bromo-4-methoxy-3-methylbenzofuran-2...)
Affinity DataIC50:  42nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50265076((R)-2-(4'-((5-bromo-4-methoxy-3-methylbenzofuran-2...)
Affinity DataIC50:  81nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50265076((R)-2-(4'-((5-bromo-4-methoxy-3-methylbenzofuran-2...)
Affinity DataIC50:  135nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50265076((R)-2-(4'-((5-bromo-4-methoxy-3-methylbenzofuran-2...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of MMP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50265076((R)-2-(4'-((5-bromo-4-methoxy-3-methylbenzofuran-2...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50265076((R)-2-(4'-((5-bromo-4-methoxy-3-methylbenzofuran-2...)
Affinity DataIC50: >7.00E+3nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50265076((R)-2-(4'-((5-bromo-4-methoxy-3-methylbenzofuran-2...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50265076((R)-2-(4'-((5-bromo-4-methoxy-3-methylbenzofuran-2...)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed