Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCollagenase 3(Homo sapiens (Human))
Zhaw Zurich University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50250159(CHEMBL4097812)
Affinity DataIC50:  89nMAssay Description:Inhibition of MMP10 (unknown origin) assessed using (5-FAM/QX) FRET peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Zhaw Zurich University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50250159(CHEMBL4097812)
Affinity DataIC50:  89nMAssay Description:Inhibition of C-terminal tagged human recombinant MMP13 catalytic domain expressed in Escherichia coli using (5-FAM/QX) FRET peptide as substrate by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-2(Homo sapiens (Human))
Zhaw Zurich University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50250159(CHEMBL4097812)
Affinity DataIC50:  243nMAssay Description:Inhibition of MMP10 (unknown origin) assessed using (5-FAM/QX) FRET peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-2(Homo sapiens (Human))
Zhaw Zurich University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50250159(CHEMBL4097812)
Affinity DataIC50:  243nMAssay Description:Inhibition of MMP10 (unknown origin) assessed using (5-FAM/QX) FRET peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed