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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Serine/threonine-protein kinase TBK1
(Homo sapiens (Human))
Gilead Sciences
US Patent
Ligand
BDBM276949
(US10072001, Example 125 | US10259811, Example 125)
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Affinity Data
IC50: 0.900nM
pH: 7.0
Assay Description:
Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Serine/threonine-protein kinase TBK1
(Homo sapiens (Human))
Gilead Sciences
US Patent
Ligand
BDBM276949
(US10072001, Example 125 | US10259811, Example 125)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.900nM
Assay Description:
Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Inhibitor of nuclear factor kappa-B kinase subunit epsilon
(Homo sapiens (Human))
Gilead Sciences
US Patent
Ligand
BDBM276949
(US10072001, Example 125 | US10259811, Example 125)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.62nM
Assay Description:
Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Inhibitor of nuclear factor kappa-B kinase subunit epsilon
(Homo sapiens (Human))
Gilead Sciences
US Patent
Ligand
BDBM276949
(US10072001, Example 125 | US10259811, Example 125)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.62nM
pH: 7.0
Assay Description:
Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI