Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetFocal adhesion kinase 1(Homo sapiens (Human))
Centaurus Biopharma

US Patent
LigandPNGBDBM245613(US9428508, 68)
Affinity DataIC50: <50nMAssay Description:To measure inhibitory activity of FAK/PYK2 inhibitors, compounds were first prepare as a 1 mM stock in 100% DMSO and 3-fold serial dilution was perfo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 2-beta(Homo sapiens (Human))
Centaurus Biopharma

US Patent
LigandPNGBDBM245613(US9428508, 68)
Affinity DataIC50: <200nMAssay Description:To measure inhibitory activity of FAK/PYK2 inhibitors, compounds were first prepare as a 1 mM stock in 100% DMSO and 3-fold serial dilution was perfo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent