Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 13 hits in this display
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
Ki: 280nMAssay Description:Inhibition of human full length recombinant His-tagged CDK2/CyclinA expressed in baculovirus using 5FAMQSPKKG-CONH2 as substrate after 60 minsMore data for this Ligand-Target Pair
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
IC50: 20nMAssay Description:Inhibition of human full length MPS1 expressed in recombinant baculovirus infected Sf9 insect cells using 5FAM-DHTGFLTEYVATRCONH2 as substrate after ...More data for this Ligand-Target Pair
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
IC50: 560nMAssay Description:Inhibition of human full length recombinant His-tagged CDK2/CyclinA expressed in baculovirus using 5FAMQSPKKG-CONH2 as substrate after 60 minsMore data for this Ligand-Target Pair
BDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)