Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Gsk

LigandBDBM27454(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-hydrox...)Copy SMILESCopy InChI

Affinity DataIC50:  2.51E+3nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair

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Ligand InfoPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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