Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Smith, Gambrell & Russell

Curated by ChEMBL

LigandBDBM50595762(CHEMBL5193680)Copy SMILESCopy InChI

Affinity DataEC50:  0.510nMAssay Description:Modulation of homozygous F508del/F508del CFTR mutant in HBE cells incubated for 18 to 24 hrs by trans-epithelial current clamp assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails PubMed
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