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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Proteasome subunit beta type-8
(Homo sapiens (Human))
Tsinghua University
Curated by
ChEMBL
Ligand
BDBM50563589
(CHEMBL4744255)
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Affinity Data
IC50: 25nM
Assay Description:
Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Proteasome subunit beta type-2
(Homo sapiens (Human))
Tsinghua University
Curated by
ChEMBL
Ligand
BDBM50563589
(CHEMBL4744255)
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Copy InChI
Affinity Data
IC50: 133nM
Assay Description:
Inhibition of 20S immunoproteasome beta 2 trypsin-like activity in human H226 cell using Z-LRR-aminoluciferin as substrate for 10 mins by fluorescenc...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-1
(Homo sapiens (Human))
Tsinghua University
Curated by
ChEMBL
Ligand
BDBM50563589
(CHEMBL4744255)
Copy SMILES
Copy InChI
Affinity Data
IC50: 418nM
Assay Description:
Inhibition of 20S immunoproteasome beta 1 caspase-like activity in human H226 cell using Z-nLPnLD-aminoluciferin as substrate for 10 mins by fluoresc...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI