Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2
(Mus musculus)
Laboratory Of Design, Synthesis, And Study Of Biologically Active Heterocycles (Heterobiolab)
Curated by
ChEMBL
Ligand
BDBM50326991
(3-((E)-4-((3,4-dimethoxyphenethyl)(methyl)amino)bu...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.72E+4nM
Assay Description:
Blockade of mouse HCN2 expressed in HEK293 cells at -120 f-current amplitude by patch-clamp electrophysiological assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4
(Homo sapiens (Human))
Laboratory Of Design, Synthesis, And Study Of Biologically Active Heterocycles (Heterobiolab)
Curated by
ChEMBL
Ligand
BDBM50326991
(3-((E)-4-((3,4-dimethoxyphenethyl)(methyl)amino)bu...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 7.23E+3nM
Assay Description:
Blockade of human HCN4 expressed in HEK293 cells at -120 f-current amplitude by patch-clamp electrophysiological assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 1
(Mus musculus)
Laboratory Of Design, Synthesis, And Study Of Biologically Active Heterocycles (Heterobiolab)
Curated by
ChEMBL
Ligand
BDBM50326991
(3-((E)-4-((3,4-dimethoxyphenethyl)(methyl)amino)bu...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 2.31E+3nM
Assay Description:
Blockade of mouse HCN1 expressed in HEK293 cells at -120 f-current amplitude by patch-clamp electrophysiological assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI