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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
22
hits in this display
Target
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: 61nM
Assay Description:
Inhibition of Axl (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
GoogleScholar
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CHEMBL
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Article
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Target
Tyrosine-protein kinase Mer
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: 126nM
Assay Description:
Inhibition of Mer (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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UniProtKB/SwissProt
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Target
Tyrosine-protein kinase receptor TYRO3
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: 270nM
Assay Description:
Inhibition of Sky (unknown origin) in presence of 60 uM ATP by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
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CHEMBL
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: 910nM
Assay Description:
Inhibition of ABL (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
UniProtKB/SwissProt
B.MOAD
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CHEMBL
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Target
Glycogen synthase kinase-3 beta
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: 1.68E+3nM
Assay Description:
Inhibition of GSK3beta (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
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KEGG
UniProtKB/SwissProt
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Target
Mitogen-activated protein kinase 1
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: 2.13E+3nM
Assay Description:
Inhibition of MAPK1/ERK2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
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CHEMBL
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PC sid
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Article
PubMed
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Target
Proto-oncogene tyrosine-protein kinase Src
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: 3.69E+3nM
Assay Description:
Inhibition of SRC (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
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Article
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Target
Insulin receptor
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: 4.65E+3nM
Assay Description:
Inhibition of INSR (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
UniProtKB/SwissProt
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Article
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Target
Hepatocyte growth factor receptor
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: 1.03E+4nM
Assay Description:
Inhibition of HGFR (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
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CHEMBL
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PC sid
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Article
PubMed
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Target
Serine/threonine-protein kinase pim-2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: 1.41E+4nM
Assay Description:
Inhibition of PIM2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
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GoogleScholar
Ligand Info
CHEMBL
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Article
PubMed
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Target
Inhibitor of nuclear factor kappa-B kinase subunit beta
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: 1.73E+4nM
Assay Description:
Inhibition of IKKbeta (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
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GoogleScholar
Ligand Info
CHEMBL
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Article
PubMed
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Target
RAC-alpha serine/threonine-protein kinase
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of AKT1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
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GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Serine/threonine-protein kinase Chk2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of CHK2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
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Target
Casein kinase I isoform delta
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of CK1delta (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
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Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of EGFR (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Inhibitor of nuclear factor kappa-B kinase subunit epsilon
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of IKKi (unknown origin)
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
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CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
MAP kinase-activated protein kinase 2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of MAPKAP-K2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of PDK1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Protein kinase C zeta type
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of PKCzeta (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Serine/threonine-protein kinase Sgk1
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of SGK (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase Chk1
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
Copy SMILES
Copy InChI
Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of CHK1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Cyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425832
(CHEMBL2312290)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of CDK2/cyclin A (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI