Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
11
hits in this display
Target
Poly [ADP-ribose] polymerase 1
(Homo sapiens (Human))
Nanjing University
Curated by
ChEMBL
Ligand
BDBM50594028
(CHEMBL5176874)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.25nM
Assay Description:
Inhibition of PARP-1 (unknown origin) using biotinylated NAD+ as substrate incubated for 45 mins in the presence of deoxy-oligonucleotide by micropla...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Poly [ADP-ribose] polymerase 1
(Homo sapiens (Human))
Nanjing University
Curated by
ChEMBL
Ligand
BDBM50594028
(CHEMBL5176874)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.25nM
Assay Description:
Inhibition of PARP1 (unknown origin) incubated for 1 hr by chemiluminescence assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Poly [ADP-ribose] polymerase 2
(Homo sapiens (Human))
Nanjing University
Curated by
ChEMBL
Ligand
BDBM50594028
(CHEMBL5176874)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.20nM
Assay Description:
Inhibition of PAPR-2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Poly [ADP-ribose] polymerase tankyrase-2
(Homo sapiens (Human))
Nanjing University
Curated by
ChEMBL
Ligand
BDBM50594028
(CHEMBL5176874)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.20nM
Assay Description:
Inhibition of TNKS2 (unknown origin) using biotin-NAD+ as substrate incubated for 1 hr in the presence of deoxy-oligonucleotide by ELISA analysis rel...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Poly [ADP-ribose] polymerase tankyrase-2
(Homo sapiens (Human))
Nanjing University
Curated by
ChEMBL
Ligand
BDBM50594028
(CHEMBL5176874)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.20nM
Assay Description:
Inhibition of tankyrase 2 (unknown origin) incubated for 1 hr by chemiluminescence based assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Poly [ADP-ribose] polymerase tankyrase-1
(Homo sapiens (Human))
Nanjing University
Curated by
ChEMBL
Ligand
BDBM50594028
(CHEMBL5176874)
Copy SMILES
Copy InChI
Affinity Data
IC50: 14nM
Assay Description:
Inhibition of TNKS1 (unknown origin) using biotin-NAD+ as substrate incubated for 1 hr in the presence of deoxy-oligonucleotide by ELISA analysis rel...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Poly [ADP-ribose] polymerase tankyrase-1
(Homo sapiens (Human))
Nanjing University
Curated by
ChEMBL
Ligand
BDBM50594028
(CHEMBL5176874)
Copy SMILES
Copy InChI
Affinity Data
IC50: 14nM
Assay Description:
Inhibition of tankyrase 1 (unknown origin) incubated for 1 hr by chemiluminescence assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Protein mono-ADP-ribosyltransferase TIPARP
(Human)
Nanjing University
Curated by
ChEMBL
Ligand
BDBM50594028
(CHEMBL5176874)
Copy SMILES
Copy InChI
Affinity Data
IC50: 15nM
Assay Description:
Inhibition of PARP-7 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Protein mono-ADP-ribosyltransferase PARP10
(Homo sapiens (Human))
Nanjing University
Curated by
ChEMBL
Ligand
BDBM50594028
(CHEMBL5176874)
Copy SMILES
Copy InChI
Affinity Data
IC50: 140nM
Assay Description:
Inhibition of PARP-10 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Protein mono-ADP-ribosyltransferase PARP12
(Homo sapiens (Human))
Nanjing University
Curated by
ChEMBL
Ligand
BDBM50594028
(CHEMBL5176874)
Copy SMILES
Copy InChI
Affinity Data
IC50: 371nM
Assay Description:
Inhibition of PARP-12 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Protein mono-ADP-ribosyltransferase PARP14
(Homo sapiens (Human))
Nanjing University
Curated by
ChEMBL
Ligand
BDBM50594028
(CHEMBL5176874)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.37E+3nM
Assay Description:
Inhibition of PARP-14 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI