Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

Target72 kDa type IV collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50101726(CHEMBL305160 | [3-(Methanesulfonyl-methyl-amino)-c...)
Affinity DataIC50:  17nMAssay Description:In vitro inhibitory concentration of the compound against Matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50101726(CHEMBL305160 | [3-(Methanesulfonyl-methyl-amino)-c...)
Affinity DataIC50:  29nMAssay Description:In vitro inhibitory concentration of the compound against Matrix metalloproteinase-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50101726(CHEMBL305160 | [3-(Methanesulfonyl-methyl-amino)-c...)
Affinity DataIC50:  560nMAssay Description:In vitro inhibitory concentration of the compound against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50101726(CHEMBL305160 | [3-(Methanesulfonyl-methyl-amino)-c...)
Affinity DataIC50:  4.66E+3nMAssay Description:In vitro inhibitory concentration of the compound against Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50101726(CHEMBL305160 | [3-(Methanesulfonyl-methyl-amino)-c...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibitory concentration of the compound against Matrix metalloproteinase-7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed