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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102472((4'-Methoxy-biphenyl-4-sulfonylamino)-[1-(3-methyl...)
Affinity DataIC50:  3.20nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50102472((4'-Methoxy-biphenyl-4-sulfonylamino)-[1-(3-methyl...)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50102472((4'-Methoxy-biphenyl-4-sulfonylamino)-[1-(3-methyl...)
Affinity DataIC50:  5.30nMAssay Description:Inhibitory activity against matrix metalloprotease-8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102472((4'-Methoxy-biphenyl-4-sulfonylamino)-[1-(3-methyl...)
Affinity DataIC50:  13.9nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102472((4'-Methoxy-biphenyl-4-sulfonylamino)-[1-(3-methyl...)
Affinity DataIC50:  14nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102472((4'-Methoxy-biphenyl-4-sulfonylamino)-[1-(3-methyl...)
Affinity DataIC50:  137nMAssay Description:In vitro inhibition of human matrix metalloprotease-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102472((4'-Methoxy-biphenyl-4-sulfonylamino)-[1-(3-methyl...)
Affinity DataIC50:  739nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102472((4'-Methoxy-biphenyl-4-sulfonylamino)-[1-(3-methyl...)
Affinity DataIC50:  4.37E+3nMAssay Description:Inhibitory activity against matrix metalloprotease-7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102472((4'-Methoxy-biphenyl-4-sulfonylamino)-[1-(3-methyl...)
Affinity DataIC50:  4.90E+3nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed