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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102473((4'-methoxy-biphenyl-4-sulfonylamino)-[1-(morpholi...)
Affinity DataIC50:  1.10nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102473((4'-methoxy-biphenyl-4-sulfonylamino)-[1-(morpholi...)
Affinity DataIC50:  1.80nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102473((4'-methoxy-biphenyl-4-sulfonylamino)-[1-(morpholi...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102473((4'-methoxy-biphenyl-4-sulfonylamino)-[1-(morpholi...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against matrix metalloprotease-8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102473((4'-methoxy-biphenyl-4-sulfonylamino)-[1-(morpholi...)
Affinity DataIC50:  3nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102473((4'-methoxy-biphenyl-4-sulfonylamino)-[1-(morpholi...)
Affinity DataIC50:  50.8nMAssay Description:In vitro inhibition of human matrix metalloprotease-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102473((4'-methoxy-biphenyl-4-sulfonylamino)-[1-(morpholi...)
Affinity DataIC50:  221nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102473((4'-methoxy-biphenyl-4-sulfonylamino)-[1-(morpholi...)
Affinity DataIC50:  1.76E+3nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102473((4'-methoxy-biphenyl-4-sulfonylamino)-[1-(morpholi...)
Affinity DataIC50:  8.57E+3nMAssay Description:Inhibitory activity against matrix metalloprotease-7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed