Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetEndothelin-1 receptor(RAT)
Merck

Curated by ChEMBL

LigandBDBM50070878(CHEMBL48881 | Sodium; (Z)-2-benzo[1,2,5]thiadiazol...)Copy SMILESCopy InChI

Affinity DataIC50:  26nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetEndothelin receptor type B(Sus scrofa)
Merck

Curated by ChEMBL

LigandBDBM50070878(CHEMBL48881 | Sodium; (Z)-2-benzo[1,2,5]thiadiazol...)Copy SMILESCopy InChI

Affinity DataIC50:  1.20E+3nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to porcine kidney (inner medulla) membranes Endothelin B receptorMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI