Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM404370(2-{(S)-3-[4-(4-Methoxy-benzoyl)-piperidin-1-yl]-2-...)
BDBM404370(2-{(S)-3-[4-(4-Methoxy-benzoyl)-piperidin-1-yl]-2-...)
IC50: 9.5nMAssay Description:The human tankyrase 1 PARP catalytic domain, TNKS1P, was cloned into a pDONR221 vector using the Invitrogen Gateway Technology. This entry clone was ...More data for this Ligand-Target Pair
BDBM404367(2-((3-(4-(4-methoxybenzoyl)piperidin-1-yl)-2-oxopy...)
IC50: 19nMAssay Description:The human tankyrase 1 PARP catalytic domain, TNKS1P, was cloned into a pDONR221 vector using the Invitrogen Gateway Technology. This entry clone was ...More data for this Ligand-Target Pair
BDBM404367(2-((3-(4-(4-methoxybenzoyl)piperidin-1-yl)-2-oxopy...)
IC50: 36nMAssay Description:The human tankyrase 1 PARP catalytic domain, TNKS1P, was cloned into a pDONR221 vector using the Invitrogen Gateway Technology. This entry clone was ...More data for this Ligand-Target Pair
BDBM404371(2-{(R)-3-[4-(4-Methoxy-benzoyl)-piperidin-1-yl]-2-...)
IC50: 390nMAssay Description:The human tankyrase 1 PARP catalytic domain, TNKS1P, was cloned into a pDONR221 vector using the Invitrogen Gateway Technology. This entry clone was ...More data for this Ligand-Target Pair
BDBM404371(2-{(R)-3-[4-(4-Methoxy-benzoyl)-piperidin-1-yl]-2-...)
IC50: 1.08E+3nMAssay Description:The human tankyrase 1 PARP catalytic domain, TNKS1P, was cloned into a pDONR221 vector using the Invitrogen Gateway Technology. This entry clone was ...More data for this Ligand-Target Pair
BDBM404371(2-{(R)-3-[4-(4-Methoxy-benzoyl)-piperidin-1-yl]-2-...)
IC50: 1.01E+4nMAssay Description:The human tankyrase 1 PARP catalytic domain, TNKS1P, was cloned into a pDONR221 vector using the Invitrogen Gateway Technology. This entry clone was ...More data for this Ligand-Target Pair
BDBM404371(2-{(R)-3-[4-(4-Methoxy-benzoyl)-piperidin-1-yl]-2-...)
IC50: >1.90E+4nMAssay Description:The human tankyrase 1 PARP catalytic domain, TNKS1P, was cloned into a pDONR221 vector using the Invitrogen Gateway Technology. This entry clone was ...More data for this Ligand-Target Pair