Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50128604((R)-3-(4-(3-(4-(3-chlorophenyl)piperazin-1-yl)prop...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibition of matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50128604((R)-3-(4-(3-(4-(3-chlorophenyl)piperazin-1-yl)prop...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of matrix metalloprotease-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50128604((R)-3-(4-(3-(4-(3-chlorophenyl)piperazin-1-yl)prop...)
Affinity DataIC50:  593nMAssay Description:In vitro inhibition of matrix metalloprotease-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed