Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetHIV-1 protease(Human immunodeficiency virus)
Umbi

Curated by ChEMBL
LigandPNGBDBM12905((5S)-N-[(1S,2R)-1-Benzyl-3-[(cyclopropylmethyl)[(4...)
Affinity DataKi:  0.575nMAssay Description:Inhibition of HIV1 protease Q7K mutant by FRET methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [491-589,Q496K](Human immunodeficiency virus type 1)
University of Massachusetts Medical School

LigandPNGBDBM12905((5S)-N-[(1S,2R)-1-Benzyl-3-[(cyclopropylmethyl)[(4...)
Affinity DataKi:  0.580nMAssay Description:HIV-1 protease inhibitor activities were determined by the fluorescence resonance energy transfer (FRET) method. The energy transfer donor (EDANS) an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHIV-1 protease(Human immunodeficiency virus)
Umbi

Curated by ChEMBL
LigandPNGBDBM12905((5S)-N-[(1S,2R)-1-Benzyl-3-[(cyclopropylmethyl)[(4...)
Affinity DataKi:  0.580nMAssay Description:Inhibition of HIV1 protease Q7K mutant by FRET methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed