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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50103994(2-[[(Benzhydryl-carbamoyl)-methyl]-(4-methoxy-benz...)
Affinity DataIC50:  0.5nMAssay Description:In vitro inhibition of human matrix metalloprotease-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Mus musculus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50078571((R)-2-[[(Benzhydryl-carbamoyl)-methyl]-(4-methoxy-...)
Affinity DataIC50:  0.5nMAssay Description:Inhibitory concentration required against matrix metalloprotease-9 (MMP-9 gelatinase B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50103994(2-[[(Benzhydryl-carbamoyl)-methyl]-(4-methoxy-benz...)
Affinity DataIC50:  2.30nMAssay Description:In vitro inhibition of human matrix metalloprotease-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Mus musculus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50078571((R)-2-[[(Benzhydryl-carbamoyl)-methyl]-(4-methoxy-...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of matrix metalloprotease-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50103994(2-[[(Benzhydryl-carbamoyl)-methyl]-(4-methoxy-benz...)
Affinity DataIC50:  3.70nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50078571((R)-2-[[(Benzhydryl-carbamoyl)-methyl]-(4-methoxy-...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of matrix metalloprotease-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078571((R)-2-[[(Benzhydryl-carbamoyl)-methyl]-(4-methoxy-...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50103994(2-[[(Benzhydryl-carbamoyl)-methyl]-(4-methoxy-benz...)
Affinity DataIC50:  4.5nMAssay Description:In vitro inhibition of human matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed