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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Stromelysin-1
(Homo sapiens (Human))
Novartis Pharmaceuticals
Ligand
BDBM13098
(CGS 27023A Analog 26 | N-hydroxy-2-[(4-methoxybenz...)
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Affinity Data
Ki: 94nM
Assay Description:
Stromelysin inhibitory activity is based on the hydrolysis of substance P by recombinant human stromelysin to generate a fragment, substance P 7-11, ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Patents
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In Depth
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Article
PubMed
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Target
Meprin A subunit beta
(Homo sapiens)
Fraunhofer Institute For Cell Therapy and Immunology Izi
Curated by
ChEMBL
Ligand
BDBM13098
(CGS 27023A Analog 26 | N-hydroxy-2-[(4-methoxybenz...)
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Affinity Data
IC50: 3.88E+4nM
Assay Description:
Inhibition of recombinant human meprin beta expressed in yeast using Abz-YVAEAPK(Dnp)G-OH as substrate by fluorescence assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI