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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50104005(1-(4-Methoxy-benzenesulfonyl)-4,4-dimethyl-3-vinyl...)
Affinity DataIC50:  138nMAssay Description:Inhibition of human matrix metalloprotease-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50104005(1-(4-Methoxy-benzenesulfonyl)-4,4-dimethyl-3-vinyl...)
Affinity DataIC50:  293nMAssay Description:Inhibition of matrix metalloprotease-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50104005(1-(4-Methoxy-benzenesulfonyl)-4,4-dimethyl-3-vinyl...)
Affinity DataIC50:  441nMAssay Description:Inhibition of matrix metalloprotease-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50104005(1-(4-Methoxy-benzenesulfonyl)-4,4-dimethyl-3-vinyl...)
Affinity DataIC50:  519nMAssay Description:Inhibition of matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50104005(1-(4-Methoxy-benzenesulfonyl)-4,4-dimethyl-3-vinyl...)
Affinity DataIC50:  2.52E+4nMAssay Description:Inhibition of human matrix metalloprotease-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed