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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098919((R)-1-Isopropyl-4-(4-methoxy-benzenesulfonyl)-7-ox...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098919((R)-1-Isopropyl-4-(4-methoxy-benzenesulfonyl)-7-ox...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of human Matrix metalloprotease-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098919((R)-1-Isopropyl-4-(4-methoxy-benzenesulfonyl)-7-ox...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of Matrix metalloprotease-8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098919((R)-1-Isopropyl-4-(4-methoxy-benzenesulfonyl)-7-ox...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098919((R)-1-Isopropyl-4-(4-methoxy-benzenesulfonyl)-7-ox...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of Matrix metalloprotease-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098919((R)-1-Isopropyl-4-(4-methoxy-benzenesulfonyl)-7-ox...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human Matrix metalloprotease-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098919((R)-1-Isopropyl-4-(4-methoxy-benzenesulfonyl)-7-ox...)
Affinity DataIC50:  369nMAssay Description:Inhibition of Matrix metalloprotease-7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed