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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

Target72 kDa type IV collagenase(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50098918((R)-1-Benzyl-3-(4-methoxy-benzenesulfonyl)-6-oxo-h...)
Affinity DataIC50:  1nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50098918((R)-1-Benzyl-3-(4-methoxy-benzenesulfonyl)-6-oxo-h...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human Matrix metalloprotease-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098918((R)-1-Benzyl-3-(4-methoxy-benzenesulfonyl)-6-oxo-h...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098918((R)-1-Benzyl-3-(4-methoxy-benzenesulfonyl)-6-oxo-h...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of Matrix metalloprotease-3More data for this Ligand-Target Pair
TargetNeutrophil collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098918((R)-1-Benzyl-3-(4-methoxy-benzenesulfonyl)-6-oxo-h...)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of Matrix metalloprotease-8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098918((R)-1-Benzyl-3-(4-methoxy-benzenesulfonyl)-6-oxo-h...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098918((R)-1-Benzyl-3-(4-methoxy-benzenesulfonyl)-6-oxo-h...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human Matrix metalloprotease-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098918((R)-1-Benzyl-3-(4-methoxy-benzenesulfonyl)-6-oxo-h...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Matrix metalloprotease-7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed