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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50118968(4-(4-Methoxy-benzenesulfonyl)-1-[2-(4-methyl-piper...)
Affinity DataIC50:  187nMAssay Description:Concentration required in vitro to inhibit Matrix metalloproteinase-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50118968(4-(4-Methoxy-benzenesulfonyl)-1-[2-(4-methyl-piper...)
Affinity DataIC50:  187nMAssay Description:Inhibition of MMP-9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50118968(4-(4-Methoxy-benzenesulfonyl)-1-[2-(4-methyl-piper...)
Affinity DataIC50:  317nMAssay Description:Concentration of the compound required in vitro to inhibit Matrix metalloproteinase-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50118968(4-(4-Methoxy-benzenesulfonyl)-1-[2-(4-methyl-piper...)
Affinity DataIC50:  317nMAssay Description:Inhibition of MMP-13 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50118968(4-(4-Methoxy-benzenesulfonyl)-1-[2-(4-methyl-piper...)
Affinity DataIC50:  808nMAssay Description:Inhibition of TACE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50118968(4-(4-Methoxy-benzenesulfonyl)-1-[2-(4-methyl-piper...)
Affinity DataIC50:  808nMAssay Description:Concentration required in vitro to inhibit TNF-alpha converting enzyme (TACE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50118968(4-(4-Methoxy-benzenesulfonyl)-1-[2-(4-methyl-piper...)
Affinity DataIC50:  4.98E+3nMAssay Description:Concentration required in vitro to inhibit Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50118968(4-(4-Methoxy-benzenesulfonyl)-1-[2-(4-methyl-piper...)
Affinity DataIC50:  4.98E+3nMAssay Description:Inhibition of MMP-1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed