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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

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TargetFree fatty acid receptor 2(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM270989(7-(4-methoxybenzenesulfonyl)-4-(3-methylpiperidin-...)
Affinity DataEC50:  41nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent