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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
24
hits in this display
Target
Serine/threonine-protein kinase 17B
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 370nM
Assay Description:
Inhibition of DRAK2 (unknown origin) using 1 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
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Target
Serine/threonine-protein kinase 17B
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 510nM
Assay Description:
Inhibition of DRAK2 (unknown origin) using 5 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
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Target
Serine/threonine-protein kinase 17B
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 530nM
Assay Description:
Inhibition of DRAK2 (unknown origin) using 10 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
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UniProtKB/SwissProt
antibodypedia
GoogleScholar
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CHEMBL
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Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 560nM
Assay Description:
Inhibition of DRAK1 (unknown origin) using 1 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
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In Depth
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Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 630nM
Assay Description:
Inhibition of DRAK1 (unknown origin) using 5 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17B
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 650nM
Assay Description:
Inhibition of DRAK2 (unknown origin) using 25 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
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In Depth
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Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 710nM
Assay Description:
Inhibition of DRAK1 (unknown origin) using 10 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17B
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 720nM
Assay Description:
Inhibition of DRAK2 (unknown origin) using 50 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17B
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 860nM
Assay Description:
Inhibition of DRAK2 (unknown origin) using 33P-ATP after 30 mins by Trilux scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 940nM
Assay Description:
Inhibition of DRAK1 (unknown origin) using 25 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17B
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 990nM
Assay Description:
Inhibition of DRAK2 (unknown origin) using 100 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17B
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.31E+3nM
Assay Description:
Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assay
More data for this Ligand-Target Pair
Target Info
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UniProtKB/SwissProt
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CHEMBL
PC cid
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PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.33E+3nM
Assay Description:
Inhibition of DRAK1 (unknown origin) using 50 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17B
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.47E+3nM
Assay Description:
Inhibition of DRAK2 (unknown origin) using 250 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.72E+3nM
Assay Description:
Inhibition of human DRAK1
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.11E+3nM
Assay Description:
Inhibition of DRAK1 (unknown origin) using 100 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
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In Depth
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Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17B
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.22E+3nM
Assay Description:
Inhibition of DRAK2 (unknown origin) using 500 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.25E+3nM
Assay Description:
Inhibition of DRAK1 (unknown origin) using 33P-ATP after 30 mins by Trilux scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.85E+3nM
Assay Description:
Inhibition of DRAK1 (unknown origin) using 250 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.91E+3nM
Assay Description:
Inhibition of DRAK1 (unknown origin) using 500 uM ATP by biochemical assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
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CHEMBL
PC cid
PC sid
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In Depth
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Article
PubMed
Copy BDB DOI
Target
Death-associated protein kinase 3
(Homo sapiens (Human))
East China Normal University
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.98E+4nM
Assay Description:
Inhibition of human DAPK3
More data for this Ligand-Target Pair
Target Info
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MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
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CHEMBL
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Copy BDB DOI
Target
Death-associated protein kinase 2
(Homo sapiens (Human))
East China Normal University
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.50E+4nM
Assay Description:
Inhibition of human DAPK2
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
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CHEMBL
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Copy BDB DOI
Target
Serine/threonine-protein kinase 17B
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
Kd: 9nM
Assay Description:
Binding affinity to DRAK2 (unknown origin) ATP site
More data for this Ligand-Target Pair
Target Info
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CHEMBL
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Copy BDB DOI
Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50024284
(CHEMBL3334979)
Copy SMILES
Copy InChI
Affinity Data
Kd: 4.90nM
Assay Description:
Binding affinity to DRAK1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
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In Depth
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PubMed
Copy BDB DOI