Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of Palermo

Curated by ChEMBL
LigandPNGBDBM50516901(CHEMBL1403454)
Affinity DataEC50:  1.50E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as iodide influx preincubated for 18 to 24 hrs follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of Palermo

Curated by ChEMBL
LigandPNGBDBM50516901(CHEMBL1403454)
Affinity DataEC50:  1.50E+4nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin incuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of Palermo

Curated by ChEMBL
LigandPNGBDBM50516901(CHEMBL1403454)
Affinity DataEC50:  3.90E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of Palermo

Curated by ChEMBL
LigandPNGBDBM50516901(CHEMBL1403454)
Affinity DataEC50:  3.90E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as iodide influx preincubated for 18 to 24 hrs followe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed