Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))TBA
LigandPNGBDBM50487746(CHEMBL2262593)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGlycogen synthase kinase-3(Homo sapiens (Human))TBA
LigandPNGBDBM50487746(CHEMBL2262593)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))TBA
LigandPNGBDBM50487746(CHEMBL2262593)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))TBA
LigandPNGBDBM50487746(CHEMBL2262593)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50487746(CHEMBL2262593)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed