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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Philochem

Curated by ChEMBL
LigandPNGBDBM50089864(CHEMBL3577702)
Affinity DataIC50:  195nMAssay Description:Inhibition of full length PARP1 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ADP-ribosyl transferase activity u...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Philochem

Curated by ChEMBL
LigandPNGBDBM50089864(CHEMBL3577702)
Affinity DataIC50:  200nMAssay Description:Inhibition of full length PARP1 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ADP-ribosyl transferase activity u...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Philochem

Curated by ChEMBL
LigandPNGBDBM50089864(CHEMBL3577702)
Affinity DataIC50:  288nMAssay Description:Inhibition of hexa-histidine tagged recombinant tankyrase 1 biotinylated catalytic domain (amino acids 1106 to 1325) (unknown origin) expressed in Es...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Philochem

Curated by ChEMBL
LigandPNGBDBM50089864(CHEMBL3577702)
Affinity DataIC50:  290nMAssay Description:Inhibition of hexa-histidine tagged recombinant tankyrase 1 biotinylated catalytic domain (amino acids 1106 to 1325) (unknown origin) expressed in Es...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Philochem

Curated by ChEMBL
LigandPNGBDBM50089864(CHEMBL3577702)
Affinity DataIC50:  330nMAssay Description:Inhibition of tankyrase 2 catalytic domain (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ADP-ribosyl transferase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Philochem

Curated by ChEMBL
LigandPNGBDBM50089864(CHEMBL3577702)
Affinity DataIC50:  331nMAssay Description:Inhibition of tankyrase 2 catalytic domain (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ADP-ribosyl transferase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
Philochem

Curated by ChEMBL
LigandPNGBDBM50089864(CHEMBL3577702)
Affinity DataIC50:  3.39E+4nMAssay Description:Inhibition of full length PARP10 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ADP-ribosyl transferase activity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
Philochem

Curated by ChEMBL
LigandPNGBDBM50089864(CHEMBL3577702)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of full length PARP10 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ADP-ribosyl transferase activity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed