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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetDual specificity protein kinase CLK4(Mus musculus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259330(CHEMBL4067420)
Affinity DataIC50:  380nMAssay Description:Inhibition of GST tagged recombinant mouse CLK4 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259330(CHEMBL4067420)
Affinity DataIC50:  930nMAssay Description:Inhibitory concentration against coagulation factor X; n=2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259330(CHEMBL4067420)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of GST tagged recombinant human DYRK2 expressed in Escherichia coli using using woodtide as substrate after 30 mins by [gamma-33P]ATP base...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259330(CHEMBL4067420)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of GST tagged recombinant mouse CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259330(CHEMBL4067420)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259330(CHEMBL4067420)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibitory concentration against dipeptidyl peptidase IVMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259330(CHEMBL4067420)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK9/cyclin T expressed in insect cells using CDK7/9-tide as substrate after 30 mins by [gamma-33P]ATP based scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259330(CHEMBL4067420)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK2/cyclin A after 30 mins by [gamma-33P]ATP based scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK3(Mus musculus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259330(CHEMBL4067420)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST tagged recombinant mouse CLK3 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259330(CHEMBL4067420)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST tagged recombinant human DYRK1B expressed in Escherichia coli using woodtide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259330(CHEMBL4067420)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 after 30 mins by [gamma-33P]ATP based scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed