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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Cystic fibrosis transmembrane conductance regulator
(Homo sapiens (Human))
University Of California Davis
Curated by
ChEMBL
Ligand
BDBM50290145
(CHEMBL2018584)
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Affinity Data
EC50: 3.70E+3nM
Assay Description:
Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Cystic fibrosis transmembrane conductance regulator
(Homo sapiens (Human))
University Of California Davis
Curated by
ChEMBL
Ligand
BDBM50290145
(CHEMBL2018584)
Copy SMILES
Copy InChI
Affinity Data
EC50: 3.72E+3nM
Assay Description:
Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI