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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Graduate School Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50175430(5-(2-METHOXYPHENYL)-2-FUROIC ACID | 5-(2-methoxyph...)
Affinity DataIC50:  558nMAssay Description:Inhibitory activity against Mn(II) form of Escherichia coli MetAPMore data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Graduate School Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50175430(5-(2-METHOXYPHENYL)-2-FUROIC ACID | 5-(2-methoxyph...)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibitory activity against Co(II) form of Escherichia coli MetAPMore data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Graduate School Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50175430(5-(2-METHOXYPHENYL)-2-FUROIC ACID | 5-(2-methoxyph...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against Ni(II) form of Escherichia coli MetAPMore data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Graduate School Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50175430(5-(2-METHOXYPHENYL)-2-FUROIC ACID | 5-(2-methoxyph...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against Fe(II) form of Escherichia coli MetAPMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50175430(5-(2-METHOXYPHENYL)-2-FUROIC ACID | 5-(2-methoxyph...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of Pin1 by PIn1 PPIase assayMore data for this Ligand-Target Pair