Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL

LigandBDBM50258787((S)-2-amino-N-(3-(5-(5-(2-methoxyphenyl)-1,3,4-oxa...)Copy SMILESCopy InChI

Affinity DataIC50:  50nMAssay Description:Inhibition of CARM1 assessed as blockade of histone H3 methylationMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI