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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetImportin subunit alpha-1(Homo sapiens (Human))
Broad Institute

Curated by PubChem BioAssay
LigandPNGBDBM75164(MLS001204421 | N-[2-(3-Cyano-5,7-dimethyl-quinolin...)
Affinity DataEC50:  4.00E+4nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California Davis

Curated by ChEMBL
LigandPNGBDBM75164(MLS001204421 | N-[2-(3-Cyano-5,7-dimethyl-quinolin...)
Affinity DataEC50:  1.10E+4nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California Davis

Curated by ChEMBL
LigandPNGBDBM75164(MLS001204421 | N-[2-(3-Cyano-5,7-dimethyl-quinolin...)
Affinity DataEC50:  1.10E+4nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed