Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University

Curated by ChEMBL

LigandBDBM50594893(CHEMBL5188771)Copy SMILESCopy InChI

Affinity DataIC50:  0.590nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathway
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails PubMed
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TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Hubei Polytechnic University

Curated by ChEMBL

LigandBDBM50594893(CHEMBL5188771)Copy SMILESCopy InChI

Affinity DataIC50:  6.5nMAssay Description:Inhibition of tankyrase 2 (unknown origin) incubated for 1 hr by chemiluminescence based assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails PubMed
Copy BDB DOI

TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Hubei Polytechnic University

Curated by ChEMBL

LigandBDBM50594893(CHEMBL5188771)Copy SMILESCopy InChI

Affinity DataIC50:  35nMAssay Description:Inhibition of tankyrase 1 (unknown origin) incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails PubMed
Copy BDB DOI