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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Endothelin-1 receptor
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50290041
(CHEMBL70203 | Pyridin-2-yl-carbamic acid 2-[6-(4-t...)
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Affinity Data
IC50: 6nM
Assay Description:
Receptor binding affinity was determined against [125I]ET1 with recombinant human ETA receptor, expressed in baculovirus-infected Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
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Target
Endothelin-1 receptor
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50290041
(CHEMBL70203 | Pyridin-2-yl-carbamic acid 2-[6-(4-t...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6nM
Assay Description:
Displacement of radioligand from ETA receptor (unknown origin) expressed in fall armyworm sf9 cell membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Endothelin-1 receptor
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50290041
(CHEMBL70203 | Pyridin-2-yl-carbamic acid 2-[6-(4-t...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6nM
Assay Description:
Displacement of radioligand from ETA receptor (unknown origin) expressed in fall armyworm sf9 cell membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Endothelin receptor type B
(Homo sapiens (Human))
Actelion Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50290041
(CHEMBL70203 | Pyridin-2-yl-carbamic acid 2-[6-(4-t...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 43nM
Assay Description:
Displacement of radioligand from ETB receptor in human placenta cell membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Endothelin receptor type B
(Homo sapiens (Human))
Actelion Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50290041
(CHEMBL70203 | Pyridin-2-yl-carbamic acid 2-[6-(4-t...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 43nM
Assay Description:
Displacement of radioligand from ETB receptor in human placenta cell membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Endothelin receptor type B
(Homo sapiens (Human))
Actelion Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50290041
(CHEMBL70203 | Pyridin-2-yl-carbamic acid 2-[6-(4-t...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 43nM
Assay Description:
Receptor binding affinity was determined against [125I]ET1 with membranes prepared from human placenta for ETB receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI