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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Casein kinase I isoform gamma-2
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50400747
(CHEMBL2203557)
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Affinity Data
IC50: 80nM
Assay Description:
Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Casein kinase I isoform alpha
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50400747
(CHEMBL2203557)
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Copy InChI
Affinity Data
IC50: 95nM
Assay Description:
Inhibition of CK1-alpha using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 8 uM ATP
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Casein kinase I isoform delta
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50400747
(CHEMBL2203557)
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Copy InChI
Affinity Data
IC50: 168nM
Assay Description:
Inhibition of CK1-delta using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 11 uM ATP
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycogen synthase kinase-3 beta
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50400747
(CHEMBL2203557)
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Copy InChI
Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of GSK3beta
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI