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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50605471(CHEMBL5181620)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human Haspin (470 to 798 residues) expressed in bacterial expression system using ARTKQTARKSTGGKAPRKQLA as substrate measur...More data for this Ligand-Target Pair
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TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50605471(CHEMBL5181620)
Affinity DataIC50:  66nMAssay Description:Inhibition of recombinant human HASPIN (470 to 798 residues) expressed in bacterial expression system in presence of ATP by kinomescan assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50605471(CHEMBL5181620)
Affinity DataIC50:  117nMAssay Description:Inhibition of human recombinant PLK3 in presence of ATP by kinomescan assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50605471(CHEMBL5181620)
Affinity DataIC50:  125nMAssay Description:Inhibition of human PLK2 in presence of ATP by kinomescan assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50605471(CHEMBL5181620)
Affinity DataIC50:  294nMAssay Description:Inhibition of human PLK1 in presence of ATP by kinomescan assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50605471(CHEMBL5181620)
Affinity DataIC50:  445nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacteria using GRSRSRSRSRSR as substrate in presence of ATP measured after 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50605471(CHEMBL5181620)
Affinity DataIC50:  578nMAssay Description:Inhibition of human DAPK3 in presence of ATP by kinomescan assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50605471(CHEMBL5181620)
Affinity DataIC50:  917nMAssay Description:Inhibition of recombinant rat DYRK1A (1 to 499 residues ) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate measured after 3...More data for this Ligand-Target Pair
In DepthDetails PubMed