Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 14 hits in this display   

TargetInterstitial collagenase(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataKi:  1nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataKi:  11nMAssay Description:Inhibition of BMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataKi:  9.10E+4nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataIC50:  9.10E+4nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed