Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50406740(CHEMBL266224)
Affinity DataKd:  200nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50406740(CHEMBL266224)
Affinity DataKd:  1.26E+4nMAssay Description:Tested for antagonist activity toward NK-3 receptor in rat portal vein against the agonist eledoisinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed