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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108523(CHEMBL3597889)
Affinity DataEC50:  5.70E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed