Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
BDBM26789(benzimidazole analog., 15 | tert-butyl (3S,4S)-3-(...)
BDBM26789(benzimidazole analog., 15 | tert-butyl (3S,4S)-3-(...)
Ki: 4.08E+3nM ΔG°: -30.8kJ/molepH: 7.5 T: 25°CAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26789(benzimidazole analog., 15 | tert-butyl (3S,4S)-3-(...)
BDBM26789(benzimidazole analog., 15 | tert-butyl (3S,4S)-3-(...)
Ki: >5.03E+3nMAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26789(benzimidazole analog., 15 | tert-butyl (3S,4S)-3-(...)
IC50: <1nMpH: 7.5 T: 25°CAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26789(benzimidazole analog., 15 | tert-butyl (3S,4S)-3-(...)
IC50: 540nMpH: 7.5 T: 25°CAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26789(benzimidazole analog., 15 | tert-butyl (3S,4S)-3-(...)
IC50: >1.00E+4nMAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair